SCHEMBL4758804

SCHEMBL4758804

CCCCOc1cc(N)nc2c1CN(c1ccccc1F)C=C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 3/20 0.39
KDM4E B2RXH2 1/20 0.37
TP53 P04637 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MCHR1 Q99705 3/20 0.36
NCF1 P14598 1/20 0.34
BACE1 P56817 3/20 0.34
CSNK1A1 P48729 1/20 0.33
CSNK1D P48730 1/20 0.33
PRKCD Q05655 1/20 0.33
PAK1 Q13153 1/20 0.33
CAMK2B Q13554 1/20 0.33
CAMK2G Q13555 1/20 0.33
CAMK2D Q13557 1/20 0.33
TAOK1 Q7L7X3 1/20 0.33
MAPK13 O15264 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788429 0.96 TLR8 (0.37) TLR8KDM4ETP53RAB9ASMN1; SMN2
SCHEMBL4790457 0.86 TLR8 (0.38) TLR8KDM4ETP53RAB9ASMN1; SMN2
SCHEMBL4108620 0.81 MCHR1 (0.38) TLR8MCHR1
SCHEMBL4796924 0.72 MEN1 (0.34) TLR8KDM4ESMN1; SMN2NCF1MAPT
SCHEMBL4786263 0.68 DCK (0.32)
SCHEMBL4812525 0.68 MAPK8 (0.37) TP53MAPK13MAPK12MAPK11MAPK14
SCHEMBL4759492 0.66 MCHR1 (0.33) TLR8MCHR1DRD2
SCHEMBL4796617 0.64 DHFR (0.34) SMN1; SMN2
SCHEMBL255559 0.62 L3MBTL1 (0.72) KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL16836380 0.62 NCF1 (0.76) TLR8CYP1A2CYP2C9CYP2C19NCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899332-A1 PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING HEPATITIS C. GILEAD SCIENCES, INC. (US) 2008-03-19 EP disclosed
WO-2006135993-A1 PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING HEPATITIS C. GILEAD SCIENCES, INC. (US) 2006-12-28 WO disclosed