SCHEMBL476048

SCHEMBL476048

C[SiH](C)CCCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
SIGMAR1 Q99720 5/20 0.48
MAOA P21397 1/20 0.48
CHRM2 P08172 1/20 0.47
HTR1A P08908 1/20 0.47
ADRA2A P08913 1/20 0.47
CHRM1 P11229 1/20 0.47
DRD1 P21728 1/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
ADRA1A P35348 1/20 0.47
OPRM1 P35372 1/20 0.47
DRD3 P35462 1/20 0.47
SLC6A3 Q01959 1/20 0.47
KCNH2 Q12809 1/20 0.47
AOC3 Q16853 1/20 0.47
MAOB P27338 1/20 0.46
HTR2A P28223 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2803699 0.93 MAOA (0.52) L3MBTL1MEN1KMT2ASIGMAR1MAOA
SCHEMBL28564556 0.91 SIGMAR1 (0.53) L3MBTL1SIGMAR1MAOAMAOB
SCHEMBL31154202 0.91 SIGMAR1 (0.53) L3MBTL1SIGMAR1MAOAMAOB
SCHEMBL476138 0.85 TP53 (0.50) L3MBTL1MAOAKCNH2AOC3MAOB
SCHEMBL17386453 0.80 TDP1 (0.52) L3MBTL1SIGMAR1MAOAADRA1ASLC6A3
SCHEMBL17453269 0.80 MEN1 (0.43) MEN1KMT2A
SCHEMBL9076218 0.79 MAOA (0.52) L3MBTL1MEN1KMT2ASIGMAR1MAOA
SCHEMBL2239331 0.79 IDO1 (0.44) L3MBTL1MEN1KMT2ASIGMAR1MAOA
SCHEMBL7560359 0.77 THRA (0.37) CHRM2ADRA2ACHRM1SLC6A2SLC6A4
SCHEMBL17206940 0.77 ESR1 (0.55) L3MBTL1KMT2ASIGMAR1CHRM2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 74 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108785142-A A kind of mascara and preparation method thereof 深圳市裕农科技股份有限公司 2018-11-13 CN claimed
CN-108409915-A A kind of Water-based polyurethane elastomer 郑细玉 2018-08-17 CN claimed
CN-108314764-A A kind of abrasion-resistance water polyurethane elastomer 郑细玉 2018-07-24 CN claimed
CN-104546561-A Three-dimensional molding wax oil powder and preparation method thereof LIXIN BIOTECH COSMETIC SHANGHAI CO LTD 2015-04-29 CN claimed
CN-104287989-A Use of polysiloxane elastomer gel in mascaras WACKER CHEMICALS CHINA CO LTD 2015-01-21 CN claimed
US-20240240086-A1 LIQUID CRYSTAL COMPOSITION, LIQUID CRYSTAL CURED LAYER, OPTICAL FILM, POLARIZING PLATE, AND IMAGE DISPLAY DEVICE FUJIFILM CORPORATION (JP) 2024-07-18 US disclosed
US-20240240086-A1 LIQUID CRYSTAL COMPOSITION, LIQUID CRYSTAL CURED LAYER, OPTICAL FILM, POLARIZING PLATE, AND IMAGE DISPLAY DEVICE FUJIFILM CORPORATION (JP) 2024-07-18 US disclosed
EP-4234643-A2 ANTIFOULING COMPOSITION Jotun A/S (NO) 2023-08-30 EP disclosed
US-20230051031-A1 MULTI-FUNCTIONAL HYBRID MATERIAL BASED ON SEPIOLITE FOR ENVIRONMENTAL RECOVERY AND BIO-REMEDIATION CONSIGLIO NAZIONALE DELLE RICERCHE (IT) 2023-02-16 US disclosed
US-20230034883-A1 MULTI-FUNCTIONAL HYBRID MATERIAL BASED ON NATURAL CLAYS FOR ENVIRONMENTAL RECOVERY AND BIO-REMEDIATION CONSIGLIO NAZIONALE DELLE RICERCHE (60%) (IT) 2023-02-02 US disclosed
EP-4076729-A1 MULTI-FUNCTIONAL HYBRID MATERIAL BASED ON NATURAL CLAYS FOR ENVIRONMENTAL RECOVERY AND BIO-REMEDIATION Consiglio Nazionale Delle Ricerche (IT) 2022-10-26 EP disclosed
EP-4076730-A1 MULTI-FUNCTIONAL HYBRID MATERIAL BASED ON SEPIOLITE FOR ENVIRONMENTAL RECOVERY AND BIO-REMEDIATION Consiglio Nazionale Delle Ricerche (IT) 2022-10-26 EP disclosed
WO-2007128550-A1 BIOCOMPATIBLE THREE DIMENSIONAL MATRIX FOR THE IMMOBILIZATION OF BIOLOGICAL SUBSTANCES LEUKOCARE AG (DE) 2007-11-15 WO disclosed
EP-1852443-A1 Biocompatible three dimensional matrix for the immobilization of biological substances Leukocare AG (DE) 2007-11-07 EP disclosed
EP-1845102-A1 NOVEL PYRIMIDINE NUCLEOSIDE COMPOUND OR ITS SALT TAIHO PHARMACEUTICAL COMPANY LIMITED (JP) 2007-10-17 EP disclosed
EP-0364344-B1 Novel peptidase inhibitors MERRELL PHARMA INC (US) 1998-05-06 EP disclosed
US-5736520-A INHIBITING CALPAIN BY ADMINISTERING A DIPEPTIDE OF THE FORMULA BENZYLCARBONYLOXYVAL-NH-CH(-R2)-CHO WHERE R2 IS THE SIDE CHAIN OF PHE; ANTICARCINOGENIC,-ARTHRITIC AND CARDIOTONIC AGENTS; COAGULANTS; STROKE MERRELL PHARMACEUTICALS INC. (US) 1998-04-07 US disclosed
EP-0363284-B1 Use of peptidase inhibitors for the preparation of medicaments useful for the treatment of strokes MERRELL PHARMA INC (US) 1997-05-14 EP disclosed
EP-0364344-A2 Novel peptidase inhibitors MERRELL PHARMACEUTICALS INC. (US) 1990-04-18 EP disclosed
EP-0363284-A2 Use of peptidase inhibitors for the preparation of medicaments useful for the treatment of strokes MERRELL PHARMACEUTICALS INC. (US) 1990-04-11 EP disclosed