SCHEMBL4760642

SCHEMBL4760642

COC(=O)Oc1c(C)c(C#N)c(N)n1-c1ccccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.40
NOTUM Q6P988 2/20 0.39
PIK3R2 O00459 1/20 0.36
GAA P10253 2/20 0.36
KDM4E B2RXH2 5/20 0.35
PIK3CD O00329 2/20 0.35
PIK3R1 P27986 2/20 0.35
APAF1 O14727 1/20 0.34
RXFP1 Q9HBX9 3/20 0.33
TSHR P16473 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33
GLA P06280 1/20 0.33
KMT2A Q03164 1/20 0.33
THRB P10828 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
PIK3CA P42336 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4891790 0.90 ALDH1A1 (0.41) ALDH1A1NOTUMGAAKDM4ETSHR
SCHEMBL4896130 0.84 ALDH1A1 (0.53) ALDH1A1GAAKDM4EPIK3CDPIK3R1
SCHEMBL4521261 0.83 ALDH1A1 (0.52) ALDH1A1NOTUMPIK3R2GAAKDM4E
SCHEMBL4894840 0.78 ALDH1A1 (0.37) ALDH1A1GAAKDM4ERXFP1TSHR
SCHEMBL4764325 0.78 L3MBTL1 (0.39) ALDH1A1NOTUMGAAKDM4ETSHR
SCHEMBL4762728 0.77 MAPT (0.39) ALDH1A1GAAKDM4ETSHRMAPT
SCHEMBL4531554 0.77 ALDH1A1 (0.48) ALDH1A1GAAKDM4ELMNAMAPT
SCHEMBL4762615 0.71 ALDH1A1 (0.45) ALDH1A1GAAKDM4ERXFP1LMNA
SCHEMBL4760669 0.71 HTT (0.44) ALDH1A1KDM4ERXFP1LMNAMAPT
SCHEMBL4721077 0.69 PARP1 (0.37) ALDH1A1NOTUMGAAKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458722-B1 PYRROLOPYRIMIDINES AS PHOSPHODIESTERASE VII INHIBITORS MERCK PATENT GMBH (DE) 2008-10-15 EP disclosed
EP-1458722-A1 PYRROLOPYRIMIDINES AS PHOSPHODIESTERASE VII INHIBITORS MERCK PATENT GmbH (DE) 2004-09-22 EP disclosed
WO-2003055882-A1 PYRROLOPYRIMIDINES AS PHOSPHODIESTERASE VII INHIBITORS MERCK PATENT GMBH (DE) 2003-07-10 WO disclosed