SCHEMBL4894840

SCHEMBL4894840

COC(=O)Oc1c(C)c(C#N)c(N)n1-c1cccs1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.37
MAPT P10636 10/20 0.36
MEN1 O00255 8/20 0.36
KMT2A Q03164 8/20 0.36
KDM4E B2RXH2 7/20 0.36
RAB9A P51151 3/20 0.36
NPC1 O15118 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HPGD P15428 2/20 0.36
HTT P42858 2/20 0.35
LMNA P02545 3/20 0.35
MITF O75030 1/20 0.35
MELK Q14680 1/20 0.34
TSHR P16473 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
RXFP1 Q9HBX9 2/20 0.33
MAPK1 P28482 2/20 0.33
HSD17B10 Q99714 4/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
USP2 O75604 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4532187 0.82 ALDH1A1 (0.49) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL4896130 0.81 ALDH1A1 (0.53) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL4760642 0.78 ALDH1A1 (0.40) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL4762728 0.70 MAPT (0.39) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL4720475 0.70 BCAT2 (0.42) ALDH1A1MAPTKMT2AKDM4EHPGD
SCHEMBL4891790 0.69 ALDH1A1 (0.41) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL6706191 0.68 ALDH1A1 (0.45) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL4760669 0.66 HTT (0.44) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL4762615 0.66 ALDH1A1 (0.45) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL4564935 0.64 ALDH1A1 (0.70) ALDH1A1MAPTMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458722-B1 PYRROLOPYRIMIDINES AS PHOSPHODIESTERASE VII INHIBITORS MERCK PATENT GMBH (DE) 2008-10-15 EP disclosed
EP-1458722-A1 PYRROLOPYRIMIDINES AS PHOSPHODIESTERASE VII INHIBITORS MERCK PATENT GmbH (DE) 2004-09-22 EP disclosed
WO-2003055882-A1 PYRROLOPYRIMIDINES AS PHOSPHODIESTERASE VII INHIBITORS MERCK PATENT GMBH (DE) 2003-07-10 WO disclosed