SCHEMBL476388

SCHEMBL476388

CN(Cc1cc(S(=O)(=O)c2ccc(F)cc2)n(-c2cccnc2F)n1)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.38
HTR6 P50406 3/20 0.37
COMT P21964 2/20 0.37
KMT2A Q03164 2/20 0.37
PTGDR2 Q9Y5Y4 5/20 0.36
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KCNA5 P22460 1/20 0.35
LIMK2 P53671 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PTGDR Q13258 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4126123 0.94 NAMPT (0.35) PKMHTR6KMT2APTGDR2
SCHEMBL3702686 0.90 HTR6 (0.40) HTR6
SCHEMBL476470 0.88 HTR6 (0.36) HTR6KMT2ALIMK2L3MBTL1
SCHEMBL476325 0.87 HTR2C (0.42) HTR6COMTKMT2APTGDR2KDM4E
SCHEMBL18258907 0.87 HTR6 (0.32) HTR6KMT2AKDM4EMAPT
SCHEMBL476326 0.86 COMT (0.36) PKMHTR6COMTKMT2APTGDR2
SCHEMBL4125764 0.85 NFE2L2 (0.40)
SCHEMBL476365 0.85 APLNR (0.35) PTGDR2KCNA5
SCHEMBL476288 0.84 COMT (0.41) PKMHTR6COMTKDM4EMAPT
SCHEMBL4135832 0.83 SLC16A3 (0.36) PKMHTR6PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2412713-B1 PYRAZOLE COMPOUND TAKEDA PHARMACEUTICAL (JP) 2016-11-30 EP disclosed
EP-2412713-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2012-02-01 EP disclosed