SCHEMBL476470

SCHEMBL476470

Cc1cccc(S(=O)(=O)c2cc(CN(C)C(=O)O)nn2-c2cccnc2F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.36
GRM1 Q13255 2/20 0.33
HRH1 P35367 1/20 0.33
GRM5 P41594 1/20 0.33
TMEM97 Q5BJF2 1/20 0.33
GRM4 Q14833 2/20 0.33
TAS2R14 Q9NYV8 1/20 0.33
NAMPT P43490 2/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33
LIMK1 P53667 1/20 0.32
LIMK2 P53671 1/20 0.32
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
KCNJ8 Q15842 1/20 0.32
ALKBH2 Q6NS38 1/20 0.32
ALKBH3 Q96Q83 1/20 0.32
FTO Q9C0B1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3702686 0.92 HTR6 (0.40) HTR6HTR2AHTR2CHTR7
SCHEMBL4126123 0.91 NAMPT (0.35) HTR6GRM1HRH1GRM5TMEM97
SCHEMBL18258907 0.90 HTR6 (0.32) HTR6NAMPTHTR2AHTR2CHTR7
SCHEMBL4125764 0.88 NFE2L2 (0.40) TAS2R14NAMPTSLC40A1
SCHEMBL476414 0.88 HTR2C (0.39) HTR6GRM1HRH1GRM5TMEM97
SCHEMBL476388 0.88 PKM (0.38) HTR6LIMK2KMT2AL3MBTL1
SCHEMBL476365 0.88 APLNR (0.35) NAMPTSLC40A1
SCHEMBL476415 0.87 HTR6 (0.35) HTR6GRM1HRH1GRM5TMEM97
SCHEMBL476363 0.86 HTR6 (0.39) HTR6GRM4NAMPTHTR2AHTR2C
SCHEMBL476471 0.84 NAMPT (0.35) HTR6GRM4NAMPTALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2412713-B1 PYRAZOLE COMPOUND TAKEDA PHARMACEUTICAL (JP) 2016-11-30 EP disclosed
EP-2412713-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2012-02-01 EP disclosed