SCHEMBL4764889

SCHEMBL4764889

CCOC(=O)OC1CCN(c2nc(CCl)nc3oc4c(c23)CCCC4)CC1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACACA Q13085 1/20 0.37
MAPT P10636 10/20 0.35
LMNA P02545 4/20 0.35
THRB P10828 2/20 0.34
KDM4E B2RXH2 5/20 0.34
ALDH1A1 P00352 4/20 0.34
HPGD P15428 4/20 0.34
NPSR1 Q6W5P4 2/20 0.34
TSHR P16473 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 2/20 0.33
POLB P06746 1/20 0.32
MAPK1 P28482 3/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32
SLC26A6 Q9BXS9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4763460 0.80 KDM4E (0.41) MAPTLMNATHRBKDM4EALDH1A1
SCHEMBL4769340 0.69 THRB (0.40) THRB
SCHEMBL1078049 0.61 ALDH1A1 (0.57) MAPTLMNAALDH1A1HSD17B10GAA
SCHEMBL4640870 0.61
SCHEMBL9330353 0.60 SCN1A (0.49) MAPTALDH1A1MEN1KMT2A
SCHEMBL8375449 0.60 ALDH1A1 (0.50) LMNATHRBALDH1A1HSD17B10GAA
SCHEMBL305155 0.60 ALDH1A1 (0.50) LMNATHRBKDM4EALDH1A1TSHR
SCHEMBL6206254 0.59 ALDH1A1 (0.51) MAPTLMNAKDM4EALDH1A1HPGD
SCHEMBL5036740 0.59 CHRM1 (0.46) MAPTLMNATHRBKDM4EALDH1A1
SCHEMBL8552607 0.58 BCHE (0.35) MAPTLMNAALDH1A1HPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432715-B1 PYRIMIDINE DERIVATIVES MERCK PATENT GMBH (DE) 2008-03-19 EP disclosed
EP-1432715-A2 PYRIMIDINE DERIVATIVES MERCK PATENT GmbH (DE) 2004-06-30 EP disclosed
WO-2003031447-A2 PYRIMIDINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-04-17 WO disclosed