SCHEMBL4767762

SCHEMBL4767762

CC1Cc2cc(F)cc(-c3cccc(Cl)c3Cl)c2O1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.51
PARP1 P09874 6/20 0.45
HTR1A P08908 5/20 0.38
BRD4 O60885 3/20 0.36
CREBBP Q92793 3/20 0.36
ALOX15 P16050 1/20 0.34
P2RX7 Q99572 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4765146 0.89 AQP1 (0.50) AQP1PARP1HTR1ABRD4CREBBP
SCHEMBL4595617 0.86 AQP1 (0.66) AQP1PARP1HTR1ABRD4CREBBP
SCHEMBL4713784 0.86 HTR1A (0.42) AQP1PARP1HTR1ABRD4CREBBP
SCHEMBL4767758 0.84 AQP1 (0.48) AQP1ALOX15P2RX7
SCHEMBL4714782 0.84 MET (0.42) AQP1PARP1HTR1ABRD4CREBBP
SCHEMBL4595103 0.82 NUDT1 (0.43) AQP1PARP1HTR1ABRD4CREBBP
SCHEMBL5185008 0.81 AQP1 (0.57) AQP1ALOX15P2RX7
SCHEMBL4219883 0.81 AQP1 (0.69) AQP1P2RX7
SCHEMBL4713102 0.80 AQP1 (0.54) AQP1PARP1HTR1ABRD4CREBBP
SCHEMBL4712234 0.80 AQP1 (0.67) AQP1PARP1HTR1ABRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879569-A2 THERAPEUTIC COMBINATIONS FOR THE TREATMENT OR PREVENTION OF PSYCHOTIC DISORDERS Wyeth (US) 2008-01-23 EP claimed
WO-2006116221-A2 THERAPEUTIC COMBINATIONS FOR THE TREATMENT OR PREVENTION OF PSYCHOTIC DISORDERS WYETH (US) 2006-11-02 WO claimed
EP-1898895-A2 TREATMENT OF DRUG ABUSE Wyeth (US) 2008-03-19 EP disclosed
EP-1871355-A1 NEW THERAPEUTIC COMBIANATIONS FOR THE TREATMENT OR PREVENTION OF DEPRESSION Wyeth (US) 2008-01-02 EP disclosed
EP-1871354-A1 TREATMENT OF PAIN Wyeth (US) 2008-01-02 EP disclosed
WO-2006116148-A2 (7-ARLYSUBSTITUTED 2, 3-DIHYDR0-1-BENZ0FURAN-2-YL) ALKYLAMINES IN THE TREATMENT' OF SUBSTANCE ABUSE WYETH (US) 2006-11-02 WO disclosed
WO-2006116149-A1 NEW THERAPEUTIC COMBIANATIONS FOR THE TREATMENT OR PREVENTION OF DEPRESSION WYETH (US) 2006-11-02 WO disclosed
WO-2006116171-A1 TREATMENT OF PAIN WYETH (US) 2006-11-02 WO disclosed