SCHEMBL4775013

SCHEMBL4775013

CCOC(=O)Oc1cc2ncn(CCC(C)(C)N)c2cn1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
POLB P06746 2/20 0.38
MAPT P10636 2/20 0.38
TNF P01375 7/20 0.36
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
LMNA P02545 1/20 0.34
CA2 P00918 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HDAC1 Q13547 1/20 0.33
F10 P00742 2/20 0.32
HPGD P15428 1/20 0.32
CDK9 P50750 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4826368 0.91 ALDH1A1 (0.38) ALDH1A1POLBMAPTTNFMTNR1A
SCHEMBL4768461 0.83 ALDH1A1 (0.38) ALDH1A1POLBMAPTTNFMTNR1A
SCHEMBL4640769 0.83 CA2 (0.44) ALDH1A1POLBMAPTTNFMTNR1A
SCHEMBL4889652 0.82 CNR2 (0.41) ALDH1A1POLBMAPTTNFLMNA
SCHEMBL4640355 0.81 MTNR1A (0.49) ALDH1A1POLBMAPTTNFMTNR1A
SCHEMBL4777107 0.79 TNF (0.36) ALDH1A1MAPTTNFCA2MEN1
SCHEMBL4913399 0.76 NPC1 (0.47) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL4893401 0.76 CNR2 (0.39) ALDH1A1POLBMAPTTNFMTNR1A
SCHEMBL4916141 0.74 NPC1 (0.48) ALDH1A1POLBMAPTTNFMTNR1A
SCHEMBL4638928 0.74 TRPM5 (0.35) ALDH1A1MAPTTNFLMNACA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945304-A2 IMIDAZO-PYRIDINE CONTAINING BETA AGONISTS, METHOD FOR PRODUCING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-23 EP disclosed
WO-2007048843-A2 IMIDAZO-PYRIDINE CONTAINING BETA AGONISTS, METHOD FOR PRODUCING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed