Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL4768481

Cc1cc(C(=O)Nc2ccc3c(c2)CCN(C2CCC2)CC3)nn1-c1ccccc1.O=C(O)C(F)(F)F

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 10/20 0.49
BCL2 P10415 1/20 0.47
RIPK1 Q13546 5/20 0.44
SLC2A1 P11166 1/20 0.44
CSF1R P07333 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
JAK3 P52333 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4777120 0.95 NPY5R (0.54) NPY5RBCL2RIPK1HRH3
Trifluoroacetic Acid SCHEMBL4774586 0.86 MAPT (0.51) SLC2A1HRH3
Trifluoroacetic Acid SCHEMBL4775487 0.86 KMT2A (0.53) SLC2A1
Trifluoroacetic Acid SCHEMBL4767895 0.85 AURKA (0.50) SLC2A1HRH3
Trifluoroacetic Acid SCHEMBL4764992 0.85 TP53 (0.51) SLC2A1HRH3
Trifluoroacetic Acid SCHEMBL4771967 0.83 SLC2A1 (0.45) SLC2A1HRH3
Trifluoroacetic Acid SCHEMBL4770119 0.83 MEN1 (0.52) SLC2A1HRH3
Trifluoroacetic Acid SCHEMBL4765180 0.82 POLB (0.52) SLC2A1HRH3
Trifluoroacetic Acid SCHEMBL4771045 0.82 RAB9A (0.53) SLC2A1
Trifluoroacetic Acid SCHEMBL4775303 0.82 ALDH1A1 (0.52) SLC2A1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1713778-B1 BENZAZEPINE DERIVATIVES AS HISTAMINE H3 ANTAGONISTS GLAXO GROUP LTD (GB) 2008-01-16 EP claimed
US-20070060566-A1 Benzazepine derivatives as histamine h3 antagonists GLAXO GROUP LIMITED (GB) 2007-03-15 US claimed
EP-1713778-B1 BENZAZEPINE DERIVATIVES AS HISTAMINE H3 ANTAGONISTS GLAXO GROUP LTD (GB) 2008-01-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070060566-A1 Benzazepine derivatives as histamine h3 antagonists HRH3, HRH4, HRH1 NPY5R 754/4885BCL2 1599/4885RIPK1 1596/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.