SCHEMBL4769975

SCHEMBL4769975

COc1cc(OC)cc(C(Cc2cnc(Cl)nc2Cl)C(=O)O)c1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ATF1 P18846 1/20 0.39
NFKB1 P19838 1/20 0.39
AKR1C3 P42330 4/20 0.38
AKR1C2 P52895 4/20 0.38
AKR1C1 Q04828 2/20 0.38
PTGS1 P23219 1/20 0.38
CCKAR P32238 12/20 0.36
AKR1B10 O60218 1/20 0.36
AKR1C4 P17516 1/20 0.36
PIN1 Q13526 1/20 0.35
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4770069 0.89 ATF1 (0.41) ATF1NFKB1PIN1KDM4EALDH1A1
SCHEMBL4764854 0.88 CCKAR (0.45) AKR1C3AKR1C2AKR1C1PTGS1CCKAR
SCHEMBL4775298 0.82 ACHE (0.41) AKR1C3AKR1C2AKR1C1PTGS1KDM4E
SCHEMBL4769954 0.81 TSPO (0.41) AKR1C3AKR1C2AKR1C1PTGS1CCKAR
SCHEMBL4767519 0.79 P4HTM (0.42) CCKARALDH1A1
SCHEMBL4770006 0.78 NFKB1 (0.47) ATF1NFKB1AKR1C3AKR1C2
SCHEMBL4765186 0.77 CCKAR (0.43) CCKARPIN1
SCHEMBL4764898 0.77 ESR1 (0.42) CCKARKDM4EALDH1A1
SCHEMBL4768134 0.77 P4HTM (0.35) AKR1C3AKR1C2CCKAR
SCHEMBL4767426 0.74 KMT2A (0.41) NFKB1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581531-B1 PYRIDINO¬2,3-D PYRIMIDINE DERIVATIVES AS SELECTIIVE KDR AND FGFR INHIBITORS HOFFMANN LA ROCHE (CH) 2008-02-27 EP claimed