SCHEMBL4770044

SCHEMBL4770044

CC(C)(C)OC(=O)N1CCC[C@H]1Nc1nc(C#N)ccc1-c1ccc(F)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
CHRM3 P20309 6/20 0.39
EED O75530 1/20 0.39
RBBP4 Q09028 1/20 0.39
SUZ12 Q15022 1/20 0.39
EZH2 Q15910 1/20 0.39
AEBP2 Q6ZN18 1/20 0.39
GPR119 Q8TDV5 3/20 0.38
USP30 Q70CQ3 2/20 0.37
UCHL1 P09936 1/20 0.37
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4764170 0.85 RORC (0.40) ALDH1A1CHRM3EEDRBBP4SUZ12
SCHEMBL4791257 0.84 ALDH1A1 (0.38) ALDH1A1CHRM3
SCHEMBL4763365 0.79 CHRM3 (0.42) ALDH1A1CHRM3
SCHEMBL4792050 0.78 CHRM3 (0.42) ALDH1A1CHRM3USP30
SCHEMBL4764117 0.77 GPR119 (0.44) CHRM3GPR119
SCHEMBL330988 0.76 ALDH1A1 (0.49) ALDH1A1USP30LMNATSHR
SCHEMBL330987 0.76 ALDH1A1 (0.49) ALDH1A1USP30LMNATSHR
SCHEMBL4762742 0.76 CHRM3 (0.42) ALDH1A1CHRM3GPR119USP30LMNA
SCHEMBL4766572 0.75 CHRM3 (0.44) ALDH1A1CHRM3LMNA
SCHEMBL4764264 0.75 ALDH1A1 (0.41) ALDH1A1CHRM3USP30LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881975-A1 N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-01-30 EP disclosed
WO-2006121218-A1 N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-11-16 WO disclosed