SCHEMBL4772732

SCHEMBL4772732

CC(C)(C)[Si](C)(C)OCCC1(c2ccccc2)CN(C(=O)O)CCO1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 1/20 0.37
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 2/20 0.33
TOP2A P11388 1/20 0.33
OPRM1 P35372 1/20 0.32
HSD11B1 P28845 2/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
HTR1A P08908 1/20 0.31
EPHX2 P34913 1/20 0.31
RORC P51449 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4158586 0.90 SCD5 (0.39) SMN1; SMN2RORC
SCHEMBL4157196 0.77 OPRD1 (0.40) HTTALDH1A1TOP2AOPRM1HSD11B1
SCHEMBL6200549 0.76 CCR5 (0.41) SLC6A2SLC6A4
SCHEMBL7499000 0.76 CCR5 (0.41) SLC6A2SLC6A4
SCHEMBL4147119 0.73 RORC (0.41) SMN1; SMN2RORC
SCHEMBL8185070 0.73 LMNA (0.38) HTTSMN1; SMN2OPRM1SLC6A2SLC6A4
SCHEMBL7500263 0.70 CCR5 (0.40) SLC6A2SLC6A4
SCHEMBL7502461 0.70 CCR5 (0.40) SLC6A2SLC6A4
SCHEMBL5895396 0.70 CYP4F2 (0.33)
SCHEMBL13926751 0.69 TOP2A (0.35) TOP2AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569931-B1 HETEROCYCLIC COMPOUNDS AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2008-10-08 EP disclosed