SCHEMBL4773433

SCHEMBL4773433

CS(=O)(=O)N(CC(N)=O)N(Cc1ccc(C(F)(F)F)nc1)C(=O)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.40
TRPM8 Q7Z2W7 11/20 0.39
NR1H2 P55055 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.36
TAS2R14 Q9NYV8 1/20 0.36
GPBAR1 Q8TDU6 2/20 0.35
PTGS2 P35354 2/20 0.34
PTGS1 P23219 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4773435 0.70 ALDH1A1 (0.48) NR1H2
SCHEMBL4777340 0.67 GAA (0.52)
SCHEMBL30394818 0.66 MAOB (0.46) MRGPRX4
SCHEMBL2310832 0.66 MAOB (0.46) MRGPRX4
SCHEMBL27654168 0.64 DAO (0.48) MRGPRX4
SCHEMBL25376011 0.63 TRPM8 (0.41) KCNH2TRPM8
SCHEMBL30481945 0.63 TRPM8 (0.41) KCNH2TRPM8
SCHEMBL17092298 0.63 KCNH2 (0.45) KCNH2TRPM8MRGPRX4
SCHEMBL4853179 0.62 PLAAT3 (0.47) MRGPRX4
SCHEMBL18256345 0.61 GRB2 (0.54) MRGPRX4PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942888-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-07-16 EP disclosed
WO-2007056078-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed