SCHEMBL4773435

SCHEMBL4773435

CS(=O)(=O)N(CC(N)=O)c1ccccc1C(=O)NCc1ccc(C(F)(F)F)nc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
HTT P42858 1/20 0.47
KMT2A Q03164 2/20 0.45
HSD17B10 Q99714 2/20 0.45
MEN1 O00255 1/20 0.45
NAMPT P43490 2/20 0.42
P2RX7 Q99572 1/20 0.41
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
GAA P10253 1/20 0.39
NR1H2 P55055 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
ALOX15 P16050 1/20 0.38
PTGER1 P34995 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4777340 0.83 GAA (0.52) GAA
SCHEMBL4776427 0.77 GAA (0.54) ALDH1A1KMT2AMEN1GAA
SCHEMBL4773432 0.74 MEN1 (0.46) ALDH1A1KMT2AHSD17B10MEN1NAMPT
SCHEMBL4773154 0.72 GAA (0.55) KMT2AMEN1GAA
SCHEMBL4881694 0.71 DGAT2 (0.40) HTTKMT2AP2RX7NR1H2TRPV1
SCHEMBL4768157 0.71 GAA (0.70) ALDH1A1NAMPTGAA
SCHEMBL4776579 0.71 GAA (0.42) HTTP2RX7GAA
SCHEMBL31236179 0.70 TRPV1 (0.51) NAMPTADORA2ATRPV1
SCHEMBL4773433 0.70 KCNH2 (0.40) NR1H2
SCHEMBL27823398 0.70 ITK (0.45) P2RX7NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942888-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-07-16 EP disclosed
WO-2007056078-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed