SCHEMBL4881694

SCHEMBL4881694

CS(=O)(=O)NCc1ccc(-c2ccccc2C(=O)NCc2ccc(C(F)(F)F)nc2)cc1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DGAT2 Q96PD7 1/20 0.40
ITK Q08881 2/20 0.40
NR1H2 P55055 1/20 0.40
TRPV1 Q8NER1 4/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
RORC P51449 1/20 0.38
PTGES O14684 3/20 0.38
P2RX7 Q99572 1/20 0.38
MTTP P55157 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4773435 0.71 ALDH1A1 (0.48) NR1H2TRPV1HTTKMT2AP2RX7
SCHEMBL27823398 0.71 ITK (0.45) ITKNR1H2P2RX7
SCHEMBL4776427 0.71 GAA (0.54) KMT2A
SCHEMBL4793709 0.70 DGAT2 (0.39) DGAT2ITKTRPV1HTTKMT2A
SCHEMBL30810190 0.70 BCAT2 (0.53) ALOX5APFEN1
Hydrochloric Acid SCHEMBL30810233 0.69 BCAT2 (0.51) ALOX5APFEN1
SCHEMBL4773432 0.69 MEN1 (0.46) ITKTRPV1KMT2AP2RX7
SCHEMBL4776425 0.68 TDP1 (0.42) DGAT2ITKKMT2A
SCHEMBL1495701 0.68 PTGS2 (0.51) ITK
SCHEMBL27823396 0.67 ITK (0.44) DGAT2ITKTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942888-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-07-16 EP disclosed
WO-2007056078-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed