SCHEMBL4774663

SCHEMBL4774663

CC(C)Oc1ccc(C(=O)NCCC(O)Cc2ccc(-c3cn(C)c(CCNC=O)n3)cc2)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CENPE Q02224 3/20 0.44
KIFC1 Q9BW19 1/20 0.38
S1PR1 P21453 6/20 0.36
CCR3 P51677 1/20 0.36
MAP4K4 O95819 2/20 0.35
MINK1 Q8N4C8 2/20 0.35
PDE10A Q9Y233 1/20 0.35
S1PR3 Q99500 1/20 0.35
S1PR5 Q9H228 1/20 0.35
WDR5 P61964 1/20 0.35
TP53 P04637 1/20 0.34
KMO O15229 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NAMPT P43490 1/20 0.34
PRKCD Q05655 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4774049 0.79 CENPE (0.37) CENPEKIFC1S1PR1CCR3MAP4K4
SCHEMBL4767596 0.79 CENPE (0.44) CENPEKIFC1S1PR1CCR3MAP4K4
SCHEMBL13707933 0.78 CENPE (0.59) CENPEKIFC1TP53ALDH1A1MAPT
SCHEMBL361204 0.76 NPC1 (0.38) CENPEKIFC1S1PR1CCR3TP53
SCHEMBL4772000 0.75 CENPE (0.37) CENPEKIFC1S1PR1S1PR3S1PR5
SCHEMBL4520166 0.74 CENPE (0.55) CENPEKIFC1S1PR1MAP4K4MINK1
SCHEMBL13161557 0.71 CENPE (0.52) CENPEKIFC1S1PR1MAP4K4MINK1
SCHEMBL13161775 0.71 CENPE (0.52) CENPEKIFC1S1PR1MAP4K4MINK1
SCHEMBL3463128 0.71 CENPE (0.52) CENPEKIFC1S1PR1MAP4K4MINK1
SCHEMBL4774986 0.71 CENPE (0.50) CENPES1PR1S1PR3S1PR5TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742907-A4 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS INC (US) 2008-01-02 EP disclosed
EP-1742907-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2007-01-17 EP disclosed
WO-2005107762-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2005-11-17 WO disclosed