SCHEMBL4765576

SCHEMBL4765576

CN1CCN(Cc2ccc(NC3=NC(=O)C(=Cc4cccc5cccnc45)S3)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHKA P35790 1/20 0.41
IKBKE Q14164 1/20 0.40
TBK1 Q9UHD2 1/20 0.40
FGFR1 P11362 1/20 0.40
CCNT1 O60563 1/20 0.39
CDK4 P11802 1/20 0.39
CCND1 P24385 1/20 0.39
CDK9 P50750 1/20 0.39
CDK6 Q00534 1/20 0.39
CDK11A Q9UQ88 1/20 0.39
JAK2 O60674 2/20 0.39
AXL P30530 4/20 0.39
MAPT P10636 1/20 0.38
WEE1 P30291 1/20 0.38
MELK Q14680 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
PKM P14618 1/20 0.37
MAPK1 P28482 1/20 0.37
JAK3 P52333 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4776063 0.86 NQO1 (0.43) FGFR1CCNT1CDK4CCND1CDK9
SCHEMBL2788133 0.84 CHKA (0.51) CHKACCNT1CDK9WEE1GRIN1
SCHEMBL2788132 0.84 CHKA (0.51) CHKACCNT1CDK9WEE1GRIN1
SCHEMBL4774422 0.81 CYP2C9 (0.36) MAPT
SCHEMBL4770645 0.74 NEK2 (0.39) CCNT1CDK9MAPTPDGFRBPDGFRA
SCHEMBL2787956 0.71 EGFR (0.52) CCNT1CDK9MAPK1TNIK
SCHEMBL2787952 0.71 EGFR (0.52) CCNT1CDK9MAPK1TNIK
SCHEMBL4765880 0.70 ROCK1 (0.43) CCNT1CDK9CDK6MAPK1JAK3
SCHEMBL4775747 0.69 GPR84 (0.38)
SCHEMBL4768194 0.69 BACE1 (0.36) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567112-B1 THIAZOLIDIN-4-ONES FOR INHIBITING hYAK3 PROTEINS SMITHKLINE BEECHAM CORP (US) 2008-10-15 EP claimed