SCHEMBL4776170

SCHEMBL4776170

c1ccc(CCCc2cc(-c3ccc(Cn4cc5ccccc5c4)cc3)nc(C3CCCCC3)n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.39
DRD2 P14416 9/20 0.37
DRD4 P21917 9/20 0.37
DRD3 P35462 8/20 0.37
PDE5A O76074 1/20 0.36
GSK3B P49841 1/20 0.36
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CDC7 O00311 1/20 0.33
ADORA1 P30542 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
PRCP P42785 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778365 0.84 PDE5A (0.40) DRD2DRD4DRD3PDE5AGSK3B
SCHEMBL14303430 0.84 PDE5A (0.40) DRD2DRD4DRD3PDE5AGSK3B
SCHEMBL4778076 0.84 PDE5A (0.40) DRD2DRD4DRD3PDE5AGSK3B
SCHEMBL4794991 0.83 ADRA1D (0.43) GSK3BMEN1ALDH1A1KMT2A
SCHEMBL4774100 0.83 NOS3 (0.42) DRD2DRD4DRD3PDE5AGSK3B
SCHEMBL4778323 0.82 NOS3 (0.43) DRD2DRD4DRD3PDE5AGSK3B
SCHEMBL4780410 0.77 NOS3 (0.44) CYP19A1DRD2DRD4DRD3PDE5A
SCHEMBL4796379 0.76 PDE5A (0.38) PDE5AKDM4EALDH1A1ADORA1NOS3
SCHEMBL4776487 0.76 PDE5A (0.38) PDE5AKDM4EALDH1A1ADORA1NOS3
SCHEMBL4780443 0.76 PDE5A (0.38) PDE5AKDM4EALDH1A1ADORA1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed