SCHEMBL4776675

SCHEMBL4776675

O=[N+]([O-])c1ccc(-c2cc(CCCc3ccccc3)nc(N3CCNCC3)n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.47
HTR1A P08908 1/20 0.46
KMT2A Q03164 1/20 0.45
ATM Q13315 1/20 0.45
SIGMAR1 Q99720 2/20 0.44
KCNJ1 P48048 1/20 0.44
KCNH2 Q12809 1/20 0.44
ADRB1 P08588 1/20 0.43
SIRT6 Q8N6T7 1/20 0.43
HTR6 P50406 1/20 0.42
ALDH1A1 P00352 2/20 0.41
CYP2C19 P33261 2/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PSD A5PKW4 2/20 0.41
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
CTSL P07711 1/20 0.41
CTSS P25774 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4774559 0.88 KMT2A (0.48) KMT2AATMSIGMAR1ALDH1A1CYP2C19
SCHEMBL4774593 0.85 ALDH1A1 (0.44) KMT2ASIGMAR1ALDH1A1CYP2C19MAPT
SCHEMBL4779650 0.75 MAPT (0.46) KMT2ASIGMAR1ALDH1A1MAPTPSD
SCHEMBL4778477 0.74 MEN1 (0.45) KMT2ASIGMAR1ALDH1A1MAPTHTT
SCHEMBL4781142 0.73 ALDH1A1 (0.48) KMT2ASIGMAR1ALDH1A1MAPTHTT
SCHEMBL4795522 0.72 PIK3CA (0.53) ATMSIGMAR1ALDH1A1MAPTHTT
SCHEMBL4774611 0.70 LTB4R (0.47) KMT2AKCNH2ALDH1A1MAPTPSD
SCHEMBL4816380 0.69 KMT2A (0.64) KMT2AATMADRB1ALDH1A1CYP2C19
SCHEMBL4776218 0.69 CYP19A1 (0.42) KMT2AALDH1A1MAPTPSD
SCHEMBL4779144 0.69 MEN1 (0.47) KMT2AATMALDH1A1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed