SCHEMBL4774593

SCHEMBL4774593

CS(=O)(=O)N1CCN(c2nc(CCCc3ccccc3)cc(-c3ccc([N+](=O)[O-])cc3)n2)CC1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
LMNA P02545 2/20 0.44
MAPT P10636 4/20 0.42
HTT P42858 3/20 0.42
CYP2C19 P33261 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HRH4 Q9H3N8 3/20 0.41
HRH1 P35367 1/20 0.41
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
POLB P06746 1/20 0.40
PSD A5PKW4 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
GBA1 P04062 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4774559 0.85 KMT2A (0.48) ALDH1A1LMNAMAPTHTTCYP2C19
SCHEMBL4776675 0.85 HTR7 (0.47) ALDH1A1MAPTHTTCYP2C19CYP1A2
SCHEMBL4778477 0.79 MEN1 (0.45) ALDH1A1LMNAMAPTHTTSIGMAR1
SCHEMBL4779650 0.74 MAPT (0.46) ALDH1A1LMNAMAPTSIGMAR1KMT2A
SCHEMBL4781142 0.71 ALDH1A1 (0.48) ALDH1A1LMNAMAPTHTTSIGMAR1
SCHEMBL4774611 0.69 LTB4R (0.47) ALDH1A1MAPTKMT2AMEN1PSD
SCHEMBL4776747 0.69 PKM (0.43) ALDH1A1LMNAMAPTCYP1A2CYP3A4
SCHEMBL4795522 0.69 PIK3CA (0.53) ALDH1A1LMNAMAPTHTTSIGMAR1
SCHEMBL4776218 0.69 CYP19A1 (0.42) ALDH1A1MAPTKMT2AMEN1POLB
SCHEMBL4779144 0.66 MEN1 (0.47) ALDH1A1LMNAMAPTCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed