SCHEMBL4778554

SCHEMBL4778554

COc1cc(Nc2cnc(C)c(-n3cc(C(=O)NCC(C)(C)C)nn3)c2)cc(C(C)(C)C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDT P30046 1/20 0.42
NR1I2 O75469 11/20 0.40
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32
TUBB3 Q13509 1/20 0.32
TUBB2A Q13885 1/20 0.32
TUBB8 Q3ZCM7 1/20 0.32
TUBA3E Q6PEY2 1/20 0.32
TUBA1A Q71U36 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778561 0.90 DDT (0.45) DDTNR1I2
SCHEMBL4779207 0.86 NR1I2 (0.38) DDTNR1I2
SCHEMBL4783994 0.85 EGFR (0.33) DDT
SCHEMBL4779766 0.84 NR1I2 (0.41) NR1I2
SCHEMBL4782091 0.83 BRAF (0.32) DDT
SCHEMBL4779088 0.82 DDR2 (0.38)
SCHEMBL4780120 0.81 DDR1 (0.35)
SCHEMBL4780940 0.81 DRD2 (0.34) DDTNR1I2DRD2DRD4DRD3
SCHEMBL4779770 0.81 NR1H4 (0.39) DDTNR1I2
SCHEMBL4783718 0.80 LMNA (0.36) DDTNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed