SCHEMBL4779433

SCHEMBL4779433

Cc1c(CN2CCC(c3c(F)cccc3Cl)CC2)c2ccccc2n1CC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 11/20 0.50
KDM4E B2RXH2 1/20 0.46
POLB P06746 1/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 3/20 0.43
AKR1A1 P14550 1/20 0.42
AKR1B1 P15121 1/20 0.42
MAPK1 P28482 1/20 0.41
STAT3 P40763 1/20 0.41
ALOX15 P16050 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4707696 0.96 PTGDR2 (0.47) PTGDR2KDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4778231 0.92 KDM4E (0.46) PTGDR2KDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4776203 0.90 KDM4E (0.46) PTGDR2KDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4778810 0.90 KDM4E (0.46) PTGDR2KDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4774108 0.90 KDM4E (0.44) PTGDR2KDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4780894 0.88 LMNA (0.47) PTGDR2KDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4773925 0.88 POLB (0.42) PTGDR2KDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4780527 0.88 SMN1; SMN2 (0.42) PTGDR2KDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4708788 0.88 KDM4E (0.44) PTGDR2KDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4780556 0.87 KDM4E (0.46) KDM4EPOLBTSHRSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008000818-A1 FLUORINATED INDOLEAMIDES USEFUL AS LIGANDS OF THE ORL-1 RECEPTOR BRANE DISCOVERY S.R.L. (IT) 2008-01-03 WO disclosed