SCHEMBL4778231

SCHEMBL4778231

Cc1c(CN2CCC(c3c(F)cccc3Cl)CC2)c2ccccc2n1CC(N)=O

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.46
TSHR P16473 2/20 0.46
POLB P06746 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PTGDR2 Q9Y5Y4 2/20 0.41
ALDH1A1 P00352 6/20 0.41
TDP1 Q9NUW8 3/20 0.40
ALOX15 P16050 1/20 0.40
ACHE P22303 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
DRD4 P21917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4776252 0.93 PTGDR2 (0.44) KDM4ETSHRPOLBSMN1; SMN2PTGDR2
SCHEMBL4781548 0.93 LMNA (0.44) KDM4ETSHRPOLBSMN1; SMN2PTGDR2
SCHEMBL4779433 0.92 PTGDR2 (0.50) KDM4ETSHRPOLBSMN1; SMN2PTGDR2
SCHEMBL4774108 0.89 KDM4E (0.44) KDM4ETSHRPOLBSMN1; SMN2PTGDR2
SCHEMBL4778810 0.89 KDM4E (0.46) KDM4ETSHRPOLBSMN1; SMN2PTGDR2
SCHEMBL4776203 0.89 KDM4E (0.46) KDM4ETSHRPOLBSMN1; SMN2PTGDR2
SCHEMBL4780894 0.88 LMNA (0.47) KDM4ETSHRPOLBSMN1; SMN2PTGDR2
Trifluoroacetic Acid SCHEMBL4707696 0.88 PTGDR2 (0.47) KDM4ETSHRPOLBSMN1; SMN2PTGDR2
SCHEMBL4780527 0.87 SMN1; SMN2 (0.42) KDM4ETSHRPOLBSMN1; SMN2PTGDR2
SCHEMBL4773925 0.87 POLB (0.42) KDM4ETSHRPOLBSMN1; SMN2PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008000818-A1 FLUORINATED INDOLEAMIDES USEFUL AS LIGANDS OF THE ORL-1 RECEPTOR BRANE DISCOVERY S.R.L. (IT) 2008-01-03 WO disclosed