SCHEMBL4779686

SCHEMBL4779686

Cc1ncc(NC(=O)c2cc(C(C)(C)C)n[nH]2)cc1-c1ccc(C(=O)NCC(C)(C)C)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 14/20 0.41
BRAF P15056 8/20 0.41
CHEK1 O14757 1/20 0.39
ADORA2A P29274 1/20 0.39
BUB1 O43683 1/20 0.38
CYP2C9 P11712 1/20 0.38
PRKACG P22612 1/20 0.38
MAPKAPK2 P49137 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
ACSL5 Q9ULC5 1/20 0.38
STK24 Q9Y6E0 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
MITF O75030 1/20 0.37
XBP1 P17861 1/20 0.37
RAB9A P51151 1/20 0.37
PAX8 Q06710 1/20 0.37
KLF5 Q13887 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4729210 0.83 TRPV1 (0.42) RAF1BRAFADORA2AMAPK14TRPV1
SCHEMBL4779963 0.81 BRAF (0.46) RAF1BRAFKDM4ERAB9A
SCHEMBL4729212 0.80 TRPV1 (0.41) RAF1BRAFADORA2AMAPK14TRPV1
SCHEMBL4729484 0.80 TRPV1 (0.41) RAF1BRAFADORA2AMAPK14TRPV1
SCHEMBL4726226 0.79 RAF1 (0.46) RAF1BRAFCYP2C9TRPV1NPC1
SCHEMBL4728383 0.79 NPC1 (0.52) RAF1BRAFADORA2ACYP2C9KDM4E
SCHEMBL4726798 0.78 RAF1 (0.42) RAF1BRAFTRPV1
SCHEMBL4725914 0.78 RAF1 (0.41) RAF1BRAFADORA2A
SCHEMBL4781066 0.78 MAPK14 (0.55) RAF1MAPK14
SCHEMBL4727602 0.78 RAF1 (0.42) RAF1BRAFADORA2AMAPK14TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed