SCHEMBL4779717

SCHEMBL4779717

CCOC(=O)CCOc1ccc(-c2ccc3nc(NCCC(C)C)ncc3c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BRAF P15056 16/20 0.43
PDE3B Q13370 2/20 0.43
PDE3A Q14432 2/20 0.43
P2RY12 Q9H244 2/20 0.43
CASR P41180 1/20 0.41
RAF1 P04049 1/20 0.40
CYSLTR2 Q9NS75 1/20 0.39
CYSLTR1 Q9Y271 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4779713 0.85 LMNA (0.40) BRAFCASRRAF1
SCHEMBL4359620 0.80 HTT (0.51)
SCHEMBL4353861 0.72 CLK4 (0.54)
SCHEMBL4351977 0.67 PDE3B (0.43) PDE3BPDE3AP2RY12CYSLTR2CYSLTR1
SCHEMBL28798228 0.67 PCSK9 (0.56) CASR
SCHEMBL3951838 0.64 L3MBTL1 (0.66)
SCHEMBL27838094 0.63 ALOX5 (0.57) PDE3BPDE3AP2RY12CYSLTR2CYSLTR1
SCHEMBL7692039 0.63 LTA4H (0.52) CYSLTR2CYSLTR1
SCHEMBL21992555 0.63 MAPT (0.60)
SCHEMBL7692040 0.63 LTA4H (0.52) CYSLTR2CYSLTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009078-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed