SCHEMBL4779845

SCHEMBL4779845

CCC(=O)NCn1cccn1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.40
THRB P10828 2/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
FDPS P14324 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
TSHR P16473 1/20 0.39
GLS O94925 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HTT P42858 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3807279 0.83 TSHR (0.47) LMNATHRBHDAC1HDAC6FDPS
SCHEMBL16001288 0.82 KMT2A (0.48) LMNATHRBMEN1KMT2ATSHR
SCHEMBL8187886 0.81 FDPS (0.42) LMNATHRBHDAC1HDAC6FDPS
SCHEMBL1259755 0.79 TDP1 (0.41) LMNATHRBHDAC1HDAC6FDPS
Hydrochloric Acid SCHEMBL8187346 0.79 FDPS (0.41) LMNATHRBHDAC1HDAC6FDPS
SCHEMBL1259224 0.77 ALDH1A1 (0.51) LMNAHDAC6MEN1KMT2AGLS
SCHEMBL27937039 0.77 KEAP1 (0.42) LMNATHRBHDAC1HDAC6MEN1
SCHEMBL7030414 0.77 NLRP3 (0.46) LMNATHRBHDAC1HDAC6MEN1
SCHEMBL8719580 0.76 MEN1 (0.43) LMNAMEN1KMT2ATSHRCYP1A2
SCHEMBL19022012 0.74 GLS (0.47) LMNATHRBHDAC1HDAC6FDPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893610-A2 ALPHA-(ARYL-OR HETEROARYL-METHYL)-BETA PIPERIDINO PROPANAMIDE COMPOUNDS AS ORL1-RECEPTOR ANTAGONISTS Pfizer, Inc. (US) 2008-03-05 EP disclosed
WO-2006134486-A2 ALPHA-(ARYL-OR HETEROARYL-METHYL)-BETA PIPERIDINO PROPANAMIDE COMPOUNDS AS ORL1-RECEPTOR ANTAGONISTS PFIZER JAPAN INC. (JP) 2006-12-21 WO disclosed