SCHEMBL4779946

SCHEMBL4779946

CCC(Oc1ccc(F)c2[nH]cc(Cc3ccc(S(=O)(=O)CC)cc3)c(=O)c12)C(=O)OC

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
RORC P51449 5/20 0.31
MKNK2 Q9HBH9 1/20 0.31
BRD4 O60885 1/20 0.31
KCNA5 P22460 1/20 0.30
TNF P01375 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4772679 0.81 MAPT (0.47) NPC1LMNATP53MAPTRAB9A
SCHEMBL4777706 0.79 NPC1 (0.43) NPC1LMNATP53MAPTRAB9A
SCHEMBL3776184 0.66 TSHR (0.36) NPC1MAPTRAB9APTGDR2SMN1; SMN2
SCHEMBL3770710 0.63 TSHR (0.37) NPC1MAPTRAB9APTGDR2SMN1; SMN2
SCHEMBL534117 0.62 P2RX3 (0.40) SMN1; SMN2
SCHEMBL168255 0.59 HPGD (0.44) RORC
SCHEMBL1550705 0.58 CLEC4M (0.58) TP53MAPT
SCHEMBL3778300 0.58 PSIP1 (0.34) MAPTSMN1; SMN2RORC
SCHEMBL21381326 0.57 SMN1; SMN2 (0.57) LMNAMAPTSMN1; SMN2
SCHEMBL23174361 0.57 ESR1 (0.45) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928457-A2 QUINOLINES AND THEIR THERAPEUTIC USE Argenta Discovery Limited (GB) 2008-06-11 EP disclosed
WO-2007036743-A2 QUINOLINES AND THEIR THERAPEUTIC USE ARGENTA DISCOVERY LIMITED (GB) 2007-04-05 WO disclosed