SCHEMBL4780502

SCHEMBL4780502

[c]1occc1CN1CCOCC1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.47
ALDH1A1 P00352 2/20 0.46
CYP2C9 P11712 1/20 0.46
ALOX15 P16050 1/20 0.46
HSD17B10 Q99714 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CXCR4 P61073 1/20 0.44
CYP2A13 Q16696 8/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.41
NCF1 P14598 1/20 0.40
POLB P06746 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
KCNJ1 P48048 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2927234 0.85 HRH3 (0.43) HRH3ALDH1A1SMN1; SMN2NCF1POLB
SCHEMBL4778748 0.83 HRH3 (0.47) HRH3ALDH1A1HTTSMN1; SMN2POLB
SCHEMBL7678459 0.80 MC4R (0.46) HRH3ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL15415811 0.70 HTT (0.51) HRH3ALDH1A1CYP2C9ALOX15HSD17B10
SCHEMBL159991 0.69 ALDH1A1 (0.53) HRH3ALDH1A1CYP2C9ALOX15HSD17B10
SCHEMBL15467001 0.69 HRH3 (0.87) HRH3ALDH1A1CYP2C9ALOX15HSD17B10
SCHEMBL27708992 0.68 ALDH1A1 (0.51) HRH3ALDH1A1CYP2C9ALOX15HSD17B10
SCHEMBL4510267 0.67 LMNA (0.42) ALDH1A1CYP2C9ALOX15HSD17B10MEN1
SCHEMBL1481687 0.67 CXCR4 (0.49) HRH3ALDH1A1CYP2C9ALOX15HSD17B10
SCHEMBL21177124 0.67 CYP2A13 (0.50) HRH3ALDH1A1CYP2C9ALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008001134-A1 1,2,3,8,9,9A-HEXAHYDRO-7H-BENZO(DE)-1,7-NAPHTHYRIDIN-7-ONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE) POLYMERASE (PARP) ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2008-01-03 WO disclosed