SCHEMBL4780940

SCHEMBL4780940

COc1c(Nc2cnc(C)c(-n3cc(C(=O)NCC(C)(C)C)nn3)c2)cc(C(C)(C)C)cc1[N+](=O)[O-]

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
DDT P30046 1/20 0.31
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
NR1I2 O75469 1/20 0.31
CA2 P00918 1/20 0.30
CA5A P35218 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780945 0.90 DDT (0.33) DRD2DRD4DRD3DDTNR1I2
SCHEMBL4783718 0.84 LMNA (0.36) DDTNR1I2
SCHEMBL4779766 0.83 NR1I2 (0.41) NR1I2
SCHEMBL4778554 0.81 DDT (0.42) DRD2DRD4DRD3DDTNR1I2
SCHEMBL4799754 0.81 MAPK14 (0.37) DDTNR1I2
SCHEMBL4780603 0.79 DRD2 (0.38) DRD2DRD4DRD3DDT
SCHEMBL4778561 0.77 DDT (0.45) DDTNR1I2
SCHEMBL4955400 0.77 BRAF (0.42)
SCHEMBL4781910 0.76 GSK3A (0.33) DDTNR1I2
SCHEMBL4783352 0.75 MAPK14 (0.36) NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed