SCHEMBL4779766

SCHEMBL4779766

COc1ccc(C(C)(C)C)cc1Nc1cnc(C)c(-n2cc(C(=O)NCC(C)(C)C)nn2)c1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 15/20 0.41
MAPK1 P28482 1/20 0.40
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4784135 0.89 CYP1A2 (0.48) NR1I2MAPK1TSHRHTT
SCHEMBL4779770 0.89 NR1H4 (0.39) NR1I2TSHR
SCHEMBL4778554 0.84 DDT (0.42) NR1I2
SCHEMBL4780940 0.83 DRD2 (0.34) NR1I2
SCHEMBL4783718 0.81 LMNA (0.36) NR1I2HTT
SCHEMBL4778561 0.79 DDT (0.45) NR1I2
SCHEMBL13843780 0.78 NR1I2 (0.41) NR1I2
SCHEMBL4779207 0.77 NR1I2 (0.38) NR1I2
SCHEMBL4783370 0.77 DDT (0.38)
SCHEMBL4799754 0.77 MAPK14 (0.37) NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed