SCHEMBL4783009

SCHEMBL4783009

COC(=O)CC(=O)c1cc(C(C)(C)C)c(OC)c(C(C)(C)C)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
KMT2A Q03164 3/20 0.49
KDM4E B2RXH2 3/20 0.49
MEN1 O00255 2/20 0.49
TNFRSF1A P19438 2/20 0.47
VCAM1 P19320 2/20 0.43
CYP3A4 P08684 1/20 0.42
TDP1 Q9NUW8 2/20 0.41
LMNA P02545 1/20 0.41
ALOX15 P16050 1/20 0.41
APEX1 P27695 1/20 0.41
MAPK1 P28482 1/20 0.41
RECQL P46063 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GAA P10253 2/20 0.38
PTGS2 P35354 2/20 0.37
ALOX5 P09917 1/20 0.37
PTGS1 P23219 1/20 0.37
TP53 P04637 1/20 0.36
KCNH2 Q12809 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4782911 0.86 MEN1 (0.46) ALDH1A1KMT2AKDM4EMEN1TNFRSF1A
SCHEMBL724655 0.85 PTGS1 (0.51) ALDH1A1KMT2AKDM4EMEN1VCAM1
SCHEMBL4783649 0.84 VCAM1 (0.39) ALDH1A1KMT2AKDM4EMEN1TNFRSF1A
SCHEMBL27871656 0.83 TNFRSF1A (0.49) ALDH1A1KMT2AKDM4EMEN1TNFRSF1A
SCHEMBL2772923 0.81 TNFRSF1A (0.48) ALDH1A1KMT2AKDM4EMEN1TNFRSF1A
SCHEMBL8947133 0.81 KDM4E (0.62) ALDH1A1KMT2AKDM4EMEN1TNFRSF1A
SCHEMBL20307621 0.80 ALDH1A1 (0.77) ALDH1A1KMT2AKDM4EMEN1TNFRSF1A
SCHEMBL5677096 0.79 TNFRSF1A (0.51) ALDH1A1KDM4ETNFRSF1ACYP3A4TDP1
SCHEMBL9729410 0.77 KMT2A (0.76) ALDH1A1KMT2AKDM4EMEN1TDP1
SCHEMBL4730730 0.77 ALDH1A1 (0.57) ALDH1A1KMT2AKDM4EMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008052288-A1 DITHIOLE COMPOUNDS AS COX INHIBITORS NEURO THERAPEUTICS LIMITED (AU) 2008-05-08 WO disclosed
WO-2008052288-A1 DITHIOLE COMPOUNDS AS COX INHIBITORS NEURO THERAPEUTICS LIMITED (AU) 2008-05-08 WO disclosed