SCHEMBL4783649

SCHEMBL4783649

COCOc1c(C(C)(C)C)cc(C(=O)CC(=O)OC)cc1C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 2/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
EGFR P00533 1/20 0.37
TNFRSF1A P19438 2/20 0.35
ALOX5 P09917 2/20 0.34
PTGS1 P23219 2/20 0.34
PTGS2 P35354 2/20 0.34
LMNA P02545 2/20 0.34
RECQL P46063 2/20 0.34
ALOX15 P16050 1/20 0.34
APEX1 P27695 1/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP3A4 P08684 1/20 0.33
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4782911 0.87 MEN1 (0.46) VCAM1MEN1KMT2AALDH1A1KDM4E
SCHEMBL4783009 0.84 ALDH1A1 (0.49) VCAM1MEN1KMT2AALDH1A1KDM4E
SCHEMBL8779698 0.83 EGFR (0.48) VCAM1ALDH1A1KDM4EEGFRTNFRSF1A
SCHEMBL8903140 0.81 TNFRSF1A (0.40) EGFRTNFRSF1APTGS2
SCHEMBL4731276 0.81 ESRRA (0.38) VCAM1EGFRTNFRSF1AALOX5PTGS1
SCHEMBL9162907 0.80 TSHR (0.42) MEN1KMT2AALDH1A1EGFRTNFRSF1A
SCHEMBL7987373 0.80 TNFRSF1A (0.37) VCAM1KDM4EEGFRTNFRSF1AALOX5
SCHEMBL724655 0.80 PTGS1 (0.51) VCAM1MEN1KMT2AALDH1A1KDM4E
SCHEMBL4728139 0.76 EGFR (0.35) VCAM1ALDH1A1KDM4EEGFRTNFRSF1A
SCHEMBL7330110 0.75 VCAM1 (0.39) VCAM1KMT2AKDM4ETNFRSF1AALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008052288-A1 DITHIOLE COMPOUNDS AS COX INHIBITORS NEURO THERAPEUTICS LIMITED (AU) 2008-05-08 WO disclosed
WO-2008052288-A1 DITHIOLE COMPOUNDS AS COX INHIBITORS NEURO THERAPEUTICS LIMITED (AU) 2008-05-08 WO disclosed