SCHEMBL4784282

SCHEMBL4784282

CC[C@H](COC)Nc1cncc(C)n1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FYN P06241 3/20 0.41
CRHR1 P34998 9/20 0.36
ADRA1A P35348 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
CDK5 Q00535 1/20 0.34
DYRK1A Q13627 1/20 0.34
CDK5R1 Q15078 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33
HCAR3 P49019 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31
ACP1 P24666 1/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4628396 0.87 FYN (0.47) FYNCRHR1CCNA2CDK2CCNA1
SCHEMBL21140560 0.77 FYN (0.38) FYNCRHR1CCNA2CDK2CCNA1
SCHEMBL5416416 0.72 FYN (0.44) FYNCRHR1CCNA2CDK2CCNA1
SCHEMBL4628001 0.71 FYN (0.46) FYNCRHR1CCNA2CDK2CCNA1
SCHEMBL15357781 0.70 TRPM8 (0.41) DYRK1AHCAR3
SCHEMBL6469022 0.70 HCAR3 (0.38) FYNCRHR1ADRA1ACCNA2CDK2
SCHEMBL6468910 0.68 FYN (0.51) FYNCRHR1CCNA2CDK2CCNA1
SCHEMBL5414326 0.68 FYN (0.46) FYNCRHR1CCNA2CDK2CCNA1
SCHEMBL14544920 0.67 CRHR1 (0.48) FYNCRHR1TAS1R3TAS1R1SYK
SCHEMBL15864503 0.67 FYN (0.58) FYNCRHR1CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008083070-A1 CRF1 RECEPTOR LIGANDS COMPRISING FUSED BICYCLIC HETEROARYL MOIETIES NEUROGEN CORPORATION (US) 2008-07-10 WO disclosed