SCHEMBL4785822

SCHEMBL4785822

OC[C@H]1Cc2ccccc2CN1c1nc(NC2CCNCC2)nc(-c2cccc(F)c2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
ROCK1 Q13464 5/20 0.36
TSHR P16473 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 2/20 0.35
MAPK1 P28482 2/20 0.35
PAK4 O96013 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
ALOX15 P16050 1/20 0.35
HIF1A Q16665 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4784054 0.90 PIK3CA (0.37) ROCK1TSHRSMN1; SMN2CYP1A2MAPK1
SCHEMBL4857757 0.87 DRD2 (0.44) SMN1; SMN2ALDH1A1LMNA
SCHEMBL4785161 0.87 CSNK1E (0.36) PIK3CBPDE4BPDE4D
SCHEMBL4784447 0.85 IDH1 (0.37) ALDH1A1TP53PDE4BPDE4D
SCHEMBL4785292 0.84 ROCK1 (0.35) ROCK1TSHRSMN1; SMN2MAPK1PAK4
SCHEMBL4784674 0.77 HRH4 (0.43) SMN1; SMN2CYP1A2ALDH1A1TP53
SCHEMBL4782277 0.74 ADORA2A (0.35) MAPK1ALDH1A1
SCHEMBL4782616 0.74 IDH1 (0.40)
SCHEMBL4782447 0.73 HRH4 (0.36) TSHRSMN1; SMN2ALDH1A1TP53PDE4B
SCHEMBL4784083 0.73 PIK3CA (0.41) CYP1A2ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed