SCHEMBL4786646

SCHEMBL4786646

COc1cccc(Sc2ccc(S(=O)(=O)N3CCc4ccc(Cl)cc4C3)c3nonc23)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.41
PPARG P37231 2/20 0.39
PPARD Q03181 2/20 0.39
PPARA Q07869 2/20 0.39
ALDH1A1 P00352 3/20 0.38
IDO1 P14902 2/20 0.38
LMNA P02545 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
AKR1C1 Q04828 1/20 0.37
HSD17B3 P37058 1/20 0.37
PKM P14618 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4787181 0.87 PKM (0.42) AKR1C3PPARGPPARDPPARAALDH1A1
SCHEMBL4788040 0.85 SMN1; SMN2 (0.41) AKR1C3ALDH1A1LMNAMEN1KMT2A
SCHEMBL4787833 0.85 AKR1C3 (0.40) AKR1C3PPARGPPARDPPARAALDH1A1
SCHEMBL4745397 0.81 KMT2A (0.43) ALDH1A1MEN1KMT2APKMMAPK1
SCHEMBL8161152 0.81 TP53 (0.45) ALDH1A1LMNAMEN1KMT2AMAPK1
SCHEMBL4788142 0.81 ESR1 (0.50) AKR1C3PPARGPPARDPPARAALDH1A1
SCHEMBL4788023 0.78 TSHR (0.43) LMNAMEN1KMT2AMAPK1
SCHEMBL4743021 0.77 ALDH1A1 (0.42) ALDH1A1LMNAMEN1KMT2AMAPK1
SCHEMBL4787281 0.77 AKR1C3 (0.47) AKR1C3PPARGPPARDPPARAALDH1A1
SCHEMBL4746067 0.76 KMT2A (0.46) ALDH1A1LMNAMEN1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008115259-A2 DERIVATIVES OF BENZOXADIAZOLE SUITABLE FOR THE TREATMENT OF CELL PROLIFERATIVE DISEASES RIGEL PHARMACEUTICALS, INC. (US) 2008-09-25 WO claimed