SCHEMBL4787181

SCHEMBL4787181

COc1ccc(Sc2ccc(S(=O)(=O)N3CCc4cc(Cl)ccc4C3)c3nonc23)cc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.42
PPARG P37231 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40
AKR1C3 P42330 4/20 0.39
AKR1C1 Q04828 1/20 0.38
LMNA P02545 2/20 0.38
ALDH1A1 P00352 2/20 0.38
PDE4B Q07343 2/20 0.37
PDE4D Q08499 1/20 0.37
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
SLC6A9 P48067 3/20 0.35
IDO1 P14902 1/20 0.34
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4786646 0.87 AKR1C3 (0.41) PKMPPARGPPARDPPARAAKR1C3
SCHEMBL4787833 0.87 AKR1C3 (0.40) PPARGPPARDPPARAAKR1C3AKR1C1
SCHEMBL4788040 0.82 SMN1; SMN2 (0.41) PKMAKR1C3AKR1C1LMNAALDH1A1
SCHEMBL8160491 0.80 ACLY (0.50) PKMLMNAALDH1A1MEN1KMT2A
SCHEMBL4746866 0.79 HTT (0.48) PKMLMNAALDH1A1MEN1KMT2A
SCHEMBL4787836 0.79 AKR1C3 (0.47) PKMAKR1C3AKR1C1LMNAALDH1A1
SCHEMBL4788418 0.76 THRB (0.47) PKMLMNAALDH1A1MEN1KMT2A
SCHEMBL4788142 0.76 ESR1 (0.50) PPARGPPARDPPARAAKR1C3AKR1C1
SCHEMBL4786482 0.76 TSHR (0.42) LMNAALDH1A1MEN1KMT2AIDO1
SCHEMBL4746102 0.75 ACLY (0.44) ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008115259-A2 DERIVATIVES OF BENZOXADIAZOLE SUITABLE FOR THE TREATMENT OF CELL PROLIFERATIVE DISEASES RIGEL PHARMACEUTICALS, INC. (US) 2008-09-25 WO claimed