SCHEMBL4736835

SCHEMBL4736835

Cn1cc(-c2nc(N)nc3c2-c2cc(NS(=O)(=O)c4ccccc4)c(Cl)cc2CC3)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 4/20 0.40
CCNB2 O95067 4/20 0.40
CCNE2 O96020 4/20 0.40
CDK1 P06493 4/20 0.40
CCNB1 P14635 4/20 0.40
CCNE1 P24864 4/20 0.40
CDK2 P24941 4/20 0.40
CDK9 P50750 4/20 0.40
CDK5 Q00535 4/20 0.40
CDK5R1 Q15078 4/20 0.40
CCNB3 Q8WWL7 4/20 0.40
DRD2 P14416 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
DRD3 P35462 1/20 0.39
HTR6 P50406 1/20 0.39
BRD4 O60885 2/20 0.38
EGLN1 Q9GZT9 1/20 0.38
FGFR1 P11362 3/20 0.36
EGFR P00533 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740757 0.89 PIK3CD (0.39) DRD2HTR2AHTR2CDRD3HTR6
SCHEMBL4737408 0.85 ADORA2A (0.40) DRD2HTR2AHTR2CDRD3HTR6
SCHEMBL4739903 0.85 PIK3CA (0.41) BRD4PIK3CDPIK3CGPIK3CAPIK3CB
SCHEMBL4740441 0.84 MEN1 (0.39) DRD2HTR2AHTR2CDRD3HTR6
SCHEMBL4786839 0.80 PIKFYVE (0.39) CCNT1CCNB2CCNE2CDK1CCNB1
SCHEMBL4739040 0.80 PIK3CD (0.35) DRD2HTR2AHTR2CDRD3HTR6
SCHEMBL4787389 0.78 ADORA2A (0.39)
SCHEMBL4787513 0.78 SLC40A1 (0.40) PIK3CDPIK3CGPIK3CAPIK3CB
SCHEMBL4740427 0.77 PLAU (0.39) DRD2HTR2AHTR2CDRD3HTR6
SCHEMBL14148284 0.76 ADORA1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed