SCHEMBL4786482

SCHEMBL4786482

COc1ccc(Sc2ccc(S(=O)(=O)N3CC(C)CC(C)C3)c3nonc23)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
GFER P55789 1/20 0.42
POLB P06746 4/20 0.41
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 3/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP2C9 P11712 1/20 0.39
LMNA P02545 2/20 0.38
THRB P10828 1/20 0.38
ALOX15 P16050 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 2/20 0.36
CYP1A2 P05177 1/20 0.35
RECQL P46063 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
IDO1 P14902 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4746166 0.90 TSHR (0.43) TSHRGFERPOLBKMT2AALDH1A1
SCHEMBL4787431 0.88 IDO1 (0.47) TSHRGFERPOLBKMT2AALDH1A1
SCHEMBL4788023 0.88 TSHR (0.43) TSHRGFERPOLBKMT2ACYP3A4
SCHEMBL4786432 0.85 TSHR (0.42) TSHRGFERPOLBKMT2AALDH1A1
SCHEMBL4746866 0.85 HTT (0.48) TSHRPOLBKMT2AALDH1A1LMNA
SCHEMBL4788418 0.84 THRB (0.47) KMT2AALDH1A1CYP3A4CYP2D6CYP2C19
SCHEMBL4746102 0.83 ACLY (0.44) POLBKMT2AALDH1A1CYP3A4CYP2D6
SCHEMBL4787200 0.82 TSHR (0.43) TSHRGFERPOLBKMT2AALDH1A1
SCHEMBL4788634 0.81 SMN1; SMN2 (0.48) TSHRPOLBKMT2AALDH1A1LMNA
SCHEMBL4743050 0.81 TSHR (0.44) TSHRGFERPOLBKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008115259-A2 DERIVATIVES OF BENZOXADIAZOLE SUITABLE FOR THE TREATMENT OF CELL PROLIFERATIVE DISEASES RIGEL PHARMACEUTICALS, INC. (US) 2008-09-25 WO claimed