SCHEMBL4794773

SCHEMBL4794773

c1ccc2[nH]c(-c3cc4nccnc4[nH]3)cc2c1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 15/20 0.60
CCNB2 O95067 15/20 0.60
CDK1 P06493 15/20 0.60
CCNB1 P14635 15/20 0.60
CCNB3 Q8WWL7 15/20 0.60
CDK5 Q00535 13/20 0.60
CDK5R1 Q15078 13/20 0.60
GSK3A P49840 9/20 0.60
CYP19A1 P11511 1/20 0.51
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
ITK Q08881 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780727 0.83 RIPK1 (0.59) GSK3BCCNB2CDK1CCNB1CCNB3
SCHEMBL4776375 0.78 RAB9A (0.50) GSK3BCYP19A1NPC1RAB9AITK
SCHEMBL374022 0.78 RAB9A (0.74) GSK3BCYP19A1NPC1RAB9AITK
SCHEMBL29631691 0.78 RAB9A (0.74) GSK3BCYP19A1NPC1RAB9AITK
SCHEMBL5179280 0.77 ITK (0.61) GSK3BCYP19A1NPC1RAB9AITK
SCHEMBL4725457 0.76 RAB9A (0.52) GSK3BCYP19A1NPC1RAB9AITK
SCHEMBL490933 0.75 CCNB2 (1.00) GSK3BCCNB2CDK1CCNB1CCNB3
SCHEMBL29912855 0.75 CCNB2 (1.00) GSK3BCCNB2CDK1CCNB1CCNB3
SCHEMBL1778158 0.74 CCNB2 (0.62) GSK3BCCNB2CDK1CCNB1CCNB3
SCHEMBL1779948 0.74 CCNB2 (0.62) GSK3BCCNB2CDK1CCNB1CCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008014249-A2 IMPROVED PREPARATIONS OF 2 -SUBSTITUTED PYRROLO [2, 3-B] PYRAZINE ( 4, 7 -DIAZAINDOLE ) COMPOUNDS SANOFI-AVENTIS (FR) 2008-01-31 WO disclosed