SCHEMBL4776375

SCHEMBL4776375

c1ccc2[nH]c(-c3cc4nc5ccccc5nc4[nH]3)cc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.50
NPC1 O15118 4/20 0.50
ITK Q08881 2/20 0.45
CYP19A1 P11511 1/20 0.45
MAPT P10636 4/20 0.45
ALDH1A1 P00352 3/20 0.45
HPGD P15428 3/20 0.45
KDM4E B2RXH2 3/20 0.45
MEN1 O00255 2/20 0.45
CASP3 P42574 2/20 0.45
KMT2A Q03164 2/20 0.45
SENP8 Q96LD8 2/20 0.45
SENP7 Q9BQF6 2/20 0.45
SENP6 Q9GZR1 2/20 0.45
KDR P35968 2/20 0.45
CHEK1 O14757 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
ESR1 P03372 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4725457 0.84 RAB9A (0.52) RAB9ANPC1ITKCYP19A1MAPT
SCHEMBL29631691 0.79 RAB9A (0.74) RAB9ANPC1ITKCYP19A1MAPT
SCHEMBL374022 0.79 RAB9A (0.74) RAB9ANPC1ITKCYP19A1MAPT
SCHEMBL4794773 0.78 GSK3B (0.60) RAB9ANPC1ITKCYP19A1GSK3B
SCHEMBL5942610 0.77 CCNB2 (0.58) RAB9ANPC1MAPTALDH1A1HPGD
SCHEMBL4780727 0.74 RIPK1 (0.59) RAB9ANPC1ITKCYP19A1GSK3B
SCHEMBL4776382 0.73 SMN1; SMN2 (0.56) RAB9ANPC1MAPTALDH1A1KDM4E
SCHEMBL924438 0.71 ESR1 (0.71) RAB9ANPC1MAPTALDH1A1HPGD
SCHEMBL31678980 0.71 ADORA3 (0.57) RAB9ANPC1ITKCYP19A1AURKA
SCHEMBL2186023 0.70 RAB9A (0.57) RAB9ANPC1ITKCYP19A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008014249-A2 IMPROVED PREPARATIONS OF 2 -SUBSTITUTED PYRROLO [2, 3-B] PYRAZINE ( 4, 7 -DIAZAINDOLE ) COMPOUNDS SANOFI-AVENTIS (FR) 2008-01-31 WO disclosed