SCHEMBL4795682

SCHEMBL4795682

CN1CCCC[C@H]1[C@@H](N)c1cccc(-c2ccncc2)c1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 8/20 0.40
ROCK1 Q13464 4/20 0.40
CHRNB4 P30926 2/20 0.38
CHRNA3 P32297 2/20 0.38
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
OPRM1 P35372 2/20 0.36
OPRD1 P41143 2/20 0.36
OPRK1 P41145 2/20 0.36
OPRL1 P41146 2/20 0.36
CHRNA7 P36544 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4782463 0.90 OPRM1 (0.44) CHRNB4CHRNA3OPRM1OPRD1OPRK1
SCHEMBL4780323 0.88 CHRNB4 (0.46) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL8220685 0.88 CHRNB4 (0.46) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL4781846 0.86 DPP4 (0.44) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL4776087 0.85 ROCK2 (0.42) ROCK2ROCK1CHRNB4CHRNA3CHRNB2
SCHEMBL4776097 0.85 ROCK2 (0.42) ROCK2ROCK1CHRNB4CHRNA3CHRNB2
SCHEMBL4795928 0.82 HTR1A (0.39) OPRM1OPRD1OPRK1OPRL1
SCHEMBL4795980 0.78 CHRNB4 (0.48) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL4776986 0.78 CHRNB4 (0.46) CHRNB4CHRNA3OPRM1OPRD1OPRK1
SCHEMBL4776989 0.78 CHRNB4 (0.46) CHRNB4CHRNA3OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008018639-A2 GLYCINE TRANSPORTER INHIBITOR TAISHO PHARMACEUTICAL CO., LTD. (JP) 2008-02-14 WO disclosed
WO-2008018639-A2 GLYCINE TRANSPORTER INHIBITOR TAISHO PHARMACEUTICAL CO., LTD. (JP) 2008-02-14 WO disclosed