SCHEMBL4780323

SCHEMBL4780323

CN1CCCC[C@H]1C(N)c1cccc(-c2cccnc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 5/20 0.46
CHRNA3 P32297 5/20 0.46
CHRNB2 P17787 5/20 0.46
CHRNA4 P43681 4/20 0.46
ALDH1A1 P00352 4/20 0.46
ACHE P22303 1/20 0.46
KDM4E B2RXH2 1/20 0.46
CHRNA7 P36544 3/20 0.45
CYP3A4 P08684 1/20 0.45
RECQL P46063 1/20 0.45
CHRNB1 P11230 2/20 0.43
CHRNB3 Q05901 2/20 0.43
CHRNA2 Q15822 2/20 0.40
PSIP1 O75475 2/20 0.40
LMNA P02545 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HTR3E A5X5Y0 1/20 0.40
TRPA1 O75762 1/20 0.40
HTR3B O95264 1/20 0.40
CHRNA1 P02708 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8220685 1.00 CHRNB4 (0.46) CHRNB4CHRNA3CHRNB2CHRNA4ALDH1A1
SCHEMBL4795980 0.88 CHRNB4 (0.48) CHRNB4CHRNA3CHRNB2CHRNA4ALDH1A1
SCHEMBL4795682 0.88 ROCK2 (0.40) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL4782463 0.85 OPRM1 (0.44) CHRNB4CHRNA3HDAC1
SCHEMBL8220552 0.81 OPRD1 (0.46) ALDH1A1KDM4ECYP3A4PSIP1BACE1
SCHEMBL4778904 0.81 OPRD1 (0.46) ALDH1A1KDM4ECYP3A4PSIP1BACE1
SCHEMBL4795928 0.81 HTR1A (0.39) ALDH1A1ACHEKDM4ECYP3A4RECQL
SCHEMBL8222689 0.76 CHRNB4 (0.48) CHRNB4CHRNA3CHRNB2CHRNA4ALDH1A1
SCHEMBL1797148 0.75 CHRNB4 (0.50) CHRNB4CHRNA3
SCHEMBL1797151 0.75 CHRNB4 (0.50) CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008018639-A2 GLYCINE TRANSPORTER INHIBITOR TAISHO PHARMACEUTICAL CO., LTD. (JP) 2008-02-14 WO disclosed