SCHEMBL480020

SCHEMBL480020

Cc1cc(C(O)(C(C)c2ccc(Oc3ccc(C(=O)O)c(F)c3)cc2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRKAB2 O43741 3/20 0.33
PRKAG1 P54619 3/20 0.33
PRKAA2 P54646 3/20 0.33
PRKAA1 Q13131 3/20 0.33
PRKAG3 Q9UGI9 3/20 0.33
PRKAG2 Q9UGJ0 3/20 0.33
PRKAB1 Q9Y478 3/20 0.33
ADRA2A P08913 1/20 0.33
CLCN2 P51788 1/20 0.33
P2RX3 P56373 1/20 0.32
MET P08581 2/20 0.31
S1PR2 O95136 2/20 0.31
PPARD Q03181 5/20 0.30
PPARA Q07869 5/20 0.30
PPARG P37231 4/20 0.30
GPR35 Q9HC97 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479931 0.94 S1PR2 (0.33) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL479915 0.93 PRKAB2 (0.33) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480052 0.91 RHEB (0.35) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480037 0.91 SCN8A (0.34) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL479197 0.90 SCN8A (0.34) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480101 0.89 MCL1 (0.35)
SCHEMBL480013 0.88 RXRB (0.35) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL480000 0.88 S1PR2 (0.33) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL479964 0.87 KDR (0.32) PPARDPPARAPPARG
SCHEMBL479741 0.86 MET (0.36) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed