Bromide

Bromide

SCHEMBL4800288

COc1ccccc1-c1nc(Nc2ccccc2)s[n+]1-c1ccccc1OC.[Br-]

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PHOSPHO1 Q8TCT1 1/20 0.49
FSCN1 Q16658 1/20 0.47
VCP P55072 1/20 0.46
HPGDS O60760 1/20 0.45
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
CYP2C19 P33261 3/20 0.41
LMNA P02545 2/20 0.41
ALOX15 P16050 2/20 0.41
HSD17B10 Q99714 2/20 0.41
JAK2 O60674 1/20 0.40
JAK3 P52333 1/20 0.40
GSK3B P49841 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
EGFR P00533 1/20 0.38
PTGS2 P35354 1/20 0.38
STK10 O94804 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL691978 0.99 FSCN1 (0.48) PHOSPHO1FSCN1VCPHPGDSCYP1A2
SCHEMBL691993 0.91 VCP (0.46) PHOSPHO1FSCN1VCPHPGDSCYP1A2
SCHEMBL691886 0.86 MAPT (0.47) VCPLMNAALOX15HSD17B10MEN1
SCHEMBL691991 0.81 FSCN1 (0.54) PHOSPHO1FSCN1LMNAMEN1KMT2A
SCHEMBL692310 0.81 FSCN1 (0.54) PHOSPHO1FSCN1VCPHPGDSLMNA
SCHEMBL693068 0.74 FSCN1 (0.45) PHOSPHO1FSCN1LMNAMEN1KMT2A
SCHEMBL19219203 0.65 CDK9 (0.57) VCPHPGDSCYP1A2CYP3A4CYP2D6
SCHEMBL12632697 0.65 FSCN1 (1.00) PHOSPHO1FSCN1LMNAMEN1KMT2A
SCHEMBL21670529 0.63 CYP1A2 (0.49) VCPHPGDSCYP1A2CYP3A4CYP2D6
SCHEMBL12297184 0.63 VCP (0.79) VCPHPGDSCYP1A2LMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7319107-B2 1,2,4-thiadiazolium derivatives as melanocortin receptor modulators JOHNSON & JOHNSON CONSUMER COMPANIES, INC. (US) 2008-01-15 US claimed