SCHEMBL479852

SCHEMBL479852

Cc1cc(C(O)(C(C)c2ccc(Oc3ccc(CC(=O)O)cc3)cc2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.40
THRB P10828 7/20 0.38
THRA P10827 6/20 0.38
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
RXRA P19793 2/20 0.35
RXRB P28702 2/20 0.35
RXRG P48443 2/20 0.35
SRD5A2 P31213 1/20 0.34
FFAR1 O14842 4/20 0.33
PPARD Q03181 2/20 0.33
PPARA Q07869 2/20 0.33
PPARG P37231 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479958 0.90 MCL1 (0.41) SMN1; SMN2THRBTHRAFFAR1PPARD
SCHEMBL480101 0.89 MCL1 (0.35) THRBTHRANR1H2NR1H3RXRA
SCHEMBL479944 0.88 RXRA (0.39) THRBTHRARXRARXRBRXRG
SCHEMBL479931 0.86 S1PR2 (0.33) THRBTHRAPPARDPPARAPPARG
SCHEMBL480020 0.86 PRKAB2 (0.33) PPARDPPARAPPARG
SCHEMBL479983 0.85 KDR (0.36) NR1H2NR1H3LMNA
SCHEMBL479912 0.84 THRB (0.35) THRBTHRALMNA
SCHEMBL480052 0.84 RHEB (0.35) THRBTHRAPPARDPPARAPPARG
SCHEMBL479790 0.84 MCL1 (0.36) THRBTHRAFFAR1PPARDPPARA
SCHEMBL479964 0.83 KDR (0.32) SMN1; SMN2THRBTHRAPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed