SCHEMBL480031

SCHEMBL480031

Cc1cc(C(O)(C(C)c2cc(Oc3ccc(Cl)c(C(=O)O)c3)ccc2Cl)C(F)(F)F)c[nH]c1=O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
TDP1 Q9NUW8 2/20 0.32
TTR P02766 1/20 0.32
PPOX P50336 1/20 0.32
MET P08581 1/20 0.32
THRA P10827 2/20 0.32
THRB P10828 2/20 0.32
PRKAG1 P54619 4/20 0.32
PRKAA2 P54646 4/20 0.32
PRKAB1 Q9Y478 4/20 0.32
PRKAB2 O43741 2/20 0.32
PRKAA1 Q13131 2/20 0.32
PRKAG3 Q9UGI9 2/20 0.32
PRKAG2 Q9UGJ0 2/20 0.32
PKM P14618 1/20 0.31
ADRB1 P08588 1/20 0.31
ADRB3 P13945 1/20 0.31
MRGPRX4 Q96LA9 1/20 0.31
GRIK1 P39086 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479741 0.94 MET (0.36) KMT2AMEN1TDP1TTRPPOX
SCHEMBL480000 0.94 S1PR2 (0.33) KMT2AMEN1TDP1TTRPPOX
SCHEMBL479915 0.92 PRKAB2 (0.33) KMT2AMEN1METTHRATHRB
SCHEMBL479970 0.90 CYP4F2 (0.37) KMT2AMEN1THRATHRBPKM
SCHEMBL479931 0.87 S1PR2 (0.33) KMT2AMEN1TDP1TTRPPOX
SCHEMBL479739 0.86 KDR (0.33) KMT2AMEN1PKMMAPT
SCHEMBL479871 0.86 MRGPRX4 (0.33) KMT2AMEN1METTHRATHRB
SCHEMBL479721 0.85 P2RX3 (0.34) MET
SCHEMBL480020 0.85 PRKAB2 (0.33) METPRKAG1PRKAA2PRKAB1PRKAB2
SCHEMBL480052 0.85 RHEB (0.35) KMT2AMEN1TDP1TTRPPOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed