SCHEMBL4807592

SCHEMBL4807592

Cc1cccc(C)c1N1CCOCC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.67
POLB P06746 1/20 0.67
LMNA P02545 1/20 0.48
PRKDC P78527 2/20 0.47
CNR2 P34972 2/20 0.47
MEN1 O00255 3/20 0.47
MAPT P10636 3/20 0.47
HTT P42858 3/20 0.47
KMT2A Q03164 3/20 0.47
KDM4E B2RXH2 2/20 0.47
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47
CYP2A13 Q16696 1/20 0.47
USP2 O75604 1/20 0.47
TP53 P04637 1/20 0.47
ALOX15 P16050 1/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3723928 0.87 ALDH1A1 (0.54) ALDH1A1POLBLMNAPRKDCCNR2
SCHEMBL15093718 0.82 ALDH1A1 (0.54) ALDH1A1POLBLMNAPRKDCCNR2
SCHEMBL17979907 0.80 ALDH1A1 (0.58) ALDH1A1POLBMAPTHTTKDM4E
SCHEMBL9424159 0.80 ALDH1A1 (0.48) ALDH1A1POLBLMNAPRKDCCNR2
SCHEMBL3723155 0.80 CYP1A2 (0.54) ALDH1A1POLBLMNAMAPTHTT
SCHEMBL15462283 0.79 ALDH1A1 (0.61) ALDH1A1POLBLMNAMEN1MAPT
SCHEMBL9424481 0.79 ALDH1A1 (0.47) ALDH1A1POLBLMNAPRKDCCNR2
SCHEMBL18027642 0.78 CRHR1 (0.49) ALDH1A1POLBLMNAMEN1MAPT
SCHEMBL21893900 0.78 ADRB1 (0.62) ALDH1A1POLBLMNAPRKDCCNR2
SCHEMBL11503875 0.77 ALDH1A1 (0.45) ALDH1A1POLBLMNAPRKDCCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022078306-A1 LARGE STERIC HINDERANCE PALLADIUM-NITROGEN-HETEROCYCLIC CARBENE COMPLEX, PREPARATION METHOD FOR SAME, APPLICATIONS OF SAME, AND SYNTHESIS METHOD FOR SONIDEGIB BASED ON SAME 中山大学 2022-04-21 WO disclosed
US-9340519-B2 Paracyclophane-based ligands, their preparation and use in catalysis JOHNSON MATTHEY PLC (GB) 2016-05-17 US disclosed
US-9340519-B2 Paracyclophane-based ligands, their preparation and use in catalysis JOHNSON MATTHEY PLC (GB) 2016-05-17 US disclosed
EP-2183259-B1 PARACYCLOPHANE-BASED LIGANDS, THEIR PREPARATION AND USE IN CATALYSIS JOHNSON MATTHEY PLC (GB) 2015-10-21 EP disclosed
US-8969624-B2 Cyclopentadienyl, indenyl or fluorenyl substituted phosphine compounds and their use in catalytic reactions EVONIK DEGUSSA GMBH (DE) 2015-03-03 US disclosed
US-8969624-B2 Cyclopentadienyl, indenyl or fluorenyl substituted phosphine compounds and their use in catalytic reactions EVONIK DEGUSSA GMBH (DE) 2015-03-03 US disclosed
EP-2057174-B1 NEW CYCLOPENTADIENYL, INDENYL OR FLUORENYL SUBSTITUTED PHOSPHINE COMPOUNDS AND THEIR USE IN CATALYTIC REACTIONS EVONIK DEGUSSA GMBH (DE) 2014-12-17 EP disclosed
US-20140330012-A1 PARACYCLOPHANE-BASED LIGANDS, THEIR PREPARATION AND USE IN CATALYSIS JOHNSON MATTHEY PUBLIC LIMITED COMPANY (GB) 2014-11-06 US disclosed
US-20140330012-A1 PARACYCLOPHANE-BASED LIGANDS, THEIR PREPARATION AND USE IN CATALYSIS JOHNSON MATTHEY PUBLIC LIMITED COMPANY (GB) 2014-11-06 US disclosed
US-8822680-B2 Paracyclophane-based ligands, their preparation and use in catalysis JOHNSON MATTHEY PLC (GB) 2014-09-02 US disclosed
US-7442800-B2 Nucleophilic heterocyclic carbene derivatives of Pd(acac)2 for cross-coupling reactions PROMERUS LLC (US) 2008-10-28 US disclosed
EP-1894938-A1 New cyclopentadienyl, indenyl or fluorenyl substituted phosphine compounds and their use in catalytic reactions Evonik Degussa GmbH (DE) 2008-03-05 EP disclosed
EP-1885669-A1 NUCLEOPHILIC HETEROCYCLIC CARBENE DERIVATIVES OF PD(ACAC)2 FOR CROSS-COUPLING REACTIONS Promerus LLC (US) 2008-02-13 EP disclosed
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
US-20060287544-A1 Nucleophilic heterocyclic carbene derivatives of Pd(acac)2 for cross-coupling reactions PROMERUS LLC (US) 2006-12-21 US disclosed
WO-2006128097-A1 NUCLEOPHILIC HETEROCYCLIC CARBENE DERIVATIVES OF PD(ACAC)2 FOR CROSS-COUPLING REACTIONS PROMERUS LLC (US) 2006-11-30 WO disclosed
EP-1097158-B1 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INST TECHNOLOGY (US) 2006-01-25 EP disclosed
EP-1354887-A1 Ligands for metals and improved metal-catalyzed processes based thereon Massachusetts Insitute of Technology (US) 2003-10-22 EP disclosed
EP-1097158-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-05-09 EP disclosed
WO-2000002887-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2000-01-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060287544-A1 Nucleophilic heterocyclic carbene derivatives of Pd(acac)2 for cross-coupling reactions NDC1, DDC, PDCD1LG2 ALDH1A1 893/4885POLB 687/4885LMNA 4016/4885
US-20140330012-A1 PARACYCLOPHANE-BASED LIGANDS, THEIR PREPARATION AND USE IN CATALYSIS CYCS, HCCS, CYC1 ALDH1A1 2283/4885POLB 541/4885LMNA 1031/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.