SCHEMBL4809484

SCHEMBL4809484

Cc1c(F)cccc1C1[CH]CN(CCCCNC(C)(C)C)CC1C(=O)c1cccc(O)c1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
TP53BP1 Q12888 4/20 0.33
DRD2 P14416 2/20 0.33
DRD3 P35462 2/20 0.33
HTR1A P08908 1/20 0.33
DRD1 P21728 1/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33
ADRA1A P35348 1/20 0.31
MET P08581 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4776847 0.87 ESRRG (0.33) DRD2DRD3HTR1ADRD1DRD4
SCHEMBL4751690 0.87 ADRB2 (0.34) ADRB2ADRB1ADRB3TP53BP1DRD2
SCHEMBL4751696 0.87 ADRB2 (0.34) ADRB2ADRB1ADRB3TP53BP1DRD2
SCHEMBL4026066 0.86 ESR1 (0.32)
SCHEMBL4751428 0.86 KIF11 (0.34) DRD2DRD3HTR1ADRD1DRD4
SCHEMBL4024173 0.84 KDM2B (0.33)
SCHEMBL4025458 0.83 NPC1 (0.36) MET
SCHEMBL4751598 0.80 MET (0.30) MET
SCHEMBL4026418 0.79 KDM1A (0.32)
SCHEMBL4021552 0.79 DRD3 (0.36) DRD2DRD3HTR1ADRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140810-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INCORPORATED (US) 2008-11-20 WO disclosed