SCHEMBL4828087

SCHEMBL4828087

C#Cc1cncc(N2CCC[C@@H](NC)C2)c1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 13/20 0.48
CHRNA3 P32297 6/20 0.47
CHRNB4 P30926 5/20 0.47
CHRNB2 P17787 5/20 0.47
CHRNA4 P43681 4/20 0.47
CHRNA1 P02708 3/20 0.47
CHRNG P07510 1/20 0.47
CHRNB1 P11230 1/20 0.47
CHRND Q07001 1/20 0.47
CHRNA2 Q15822 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4830391 1.00 HRH4 (0.48) HRH4CHRNA3CHRNB4CHRNB2CHRNA4
SCHEMBL4824732 0.87 CHRNB2 (0.54) HRH4CHRNA3CHRNB4CHRNB2CHRNA4
SCHEMBL4823979 0.87 CHRNB2 (0.54) HRH4CHRNA3CHRNB4CHRNB2CHRNA4
SCHEMBL4827864 0.81 CHRNA3 (0.46) HRH4CHRNA3CHRNB4CHRNB2CHRNA4
SCHEMBL4828940 0.81 CHRNA3 (0.46) HRH4CHRNA3CHRNB4CHRNB2CHRNA4
SCHEMBL4825453 0.80 ROCK2 (0.52) HRH4
SCHEMBL4819971 0.80 ROCK2 (0.52) HRH4
SCHEMBL29108032 0.78 CHRNB2 (0.47) CHRNA3CHRNB4CHRNB2CHRNA4CHRNA1
SCHEMBL29108020 0.78 CHRNB2 (0.47) CHRNA3CHRNB4CHRNB2CHRNA4CHRNA1
SCHEMBL30665748 0.78 CHRNB2 (0.47) CHRNA3CHRNB4CHRNB2CHRNA4CHRNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7332504-B2 Heterocyclic substituted aminoazacycles useful as central nervous system agents ABBOTT LABORATORIES (US) 2008-02-19 US claimed
US-7332504-B2 Heterocyclic substituted aminoazacycles useful as central nervous system agents ABBOTT LABORATORIES (US) 2008-02-19 US disclosed